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Target
X-box-binding protein 1
Ligand
BDBM68017
Substrate
n/a
Meas. Tech.
XBP1 DR counterscreen for CHOP
IC50
160±n/a nM
Citation
 PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay (2011)[AID] 
Target
Name:
X-box-binding protein 1
Synonyms:
TREB5 | XBP1 | XBP1_HUMAN | XBP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28704.14
Organism:
Homo sapiens (Human)
Description:
gi_47678753
Residue:
261
Sequence:
MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARKRQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLREKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQLSPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVPYQPPFLCQWGRHQPSWKPLMN
  
Inhibitor
Name:
BDBM68017
Synonyms:
2-(4-methylanilino)-N-[(3-phenoxyphenyl)methylideneamino]acetamide | 2-[(4-methylphenyl)amino]-N'-[(1E)-(3-phenoxyphenyl)methylene]acetohydrazide | 2-[(4-methylphenyl)amino]-N-[(3-phenoxyphenyl)methylideneamino]ethanamide | MLS000586151 | N-[(3-phenoxybenzylidene)amino]-2-(p-toluidino)acetamide | SMR000204514 | cid_1520328
Type:
Small organic molecule
Emp. Form.:
C22H21N3O2
Mol. Mass.:
359.421
SMILES:
Cc1ccc(NCC(=O)NN=Cc2cccc(Oc3ccccc3)c2)cc1
Structure:
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