Reaction Details Report a problem with these data
Target
DNA damage-inducible transcript 3 protein
Ligand
BDBM68017
Substrate
n/a
Meas. Tech.
CHOP dose-response primary assay
IC50
360±n/a nM
Citation
 PubChem, PC CHOP dose-response primary assay PubChem Bioassay (2011)[AID] 
Target
Name:
DNA damage-inducible transcript 3 protein
Synonyms:
Chop | Chop10 | DDIT3_MOUSE | Ddit3 | Gadd153
Type:
Enzyme Catalytic Domain
Mol. Mass.:
19175.17
Organism:
Mus musculus
Description:
gi_160707929
Residue:
168
Sequence:
MAAESLPFTLETVSSWELEAWYEDLQEVLSSDEIGGTYISSPGNEEEESKTFTTLDPASLAWLTEEPGPTEVTRTSQSPRSPDSSQSSMAQEEEEEEQGRTRKRKQSGQCPARPGKQRMKEKEQENERKVAQLAEENERLKQEIERLTREVETTRRALIDRMVSLHQA
  
Inhibitor
Name:
BDBM68017
Synonyms:
2-(4-methylanilino)-N-[(3-phenoxyphenyl)methylideneamino]acetamide | 2-[(4-methylphenyl)amino]-N'-[(1E)-(3-phenoxyphenyl)methylene]acetohydrazide | 2-[(4-methylphenyl)amino]-N-[(3-phenoxyphenyl)methylideneamino]ethanamide | MLS000586151 | N-[(3-phenoxybenzylidene)amino]-2-(p-toluidino)acetamide | SMR000204514 | cid_1520328
Type:
Small organic molecule
Emp. Form.:
C22H21N3O2
Mol. Mass.:
359.421
SMILES:
Cc1ccc(NCC(=O)NN=Cc2cccc(Oc3ccccc3)c2)cc1
Structure:
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