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Target
Kappa-type opioid receptor [1-7]
Ligand
BDBM42323
Substrate
n/a
Meas. Tech.
Late-stage radioligand binding dose response assay to identify inhibitors of NADPH oxidase 1 (NOX1): PDSP screen Ki Set 2
Ki
>10000±n/a nM
Citation
 PubChem, PC Late-stage radioligand binding dose response assay to identify inhibitors of NADPH oxidase 1 (NOX1): PDSP screen Ki Set 2 PubChem Bioassay (2011)[AID] 
Target
Name:
Kappa-type opioid receptor [1-7]
Synonyms:
OPRK | OPRK1 | OPRK_HUMAN | kappa opioid receptor | kappa opioid receptor [Homo sapiens]
Type:
Enzyme Catalytic Domain
Mol. Mass.:
801.93
Organism:
Homo sapiens (Human)
Description:
gi_39986053
Residue:
7
Sequence:
MDSPIQI
  
Inhibitor
Name:
BDBM42323
Synonyms:
1-(10H-phenothiazin-2-yl)ethanone | MLS000047624 | SMR000033635 | cid_81131
Type:
Small organic molecule
Emp. Form.:
C14H11NOS
Mol. Mass.:
241.308
SMILES:
CC(=O)c1ccc2Sc3ccccc3Nc2c1
Structure:
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