Reaction Details Report a problem with these data
Target
5-hydroxytryptamine 1D receptor
Ligand
BDBM21395
Substrate
n/a
Ki
3200±n/a nM
Comments
PDSP_1014
Citation
 Leonhardt, S; Herrick-Davis, K; Titeler, M Detection of a novel serotonin receptor subtype (5-HT1E) in human brain: interaction with a GTP-binding protein. J Neurochem 53:465-71 (1989) [PubMed]  Article 
Target
Name:
5-hydroxytryptamine 1D receptor
Synonyms:
5-hydroxytryptamine 1D receptor (5HT1D) | HTR1D
Type:
Protein
Mol. Mass.:
12731.52
Organism:
Bos taurus (Bovine)
Description:
Q8MI13
Residue:
119
Sequence:
SNRSLNATATQGAWDPGTLQALKIALVVLLSIITLATVLSNAFVLTTIFLTRKLHTPANCLIGSLAMTDLLVSILVMPISIAYTTTHTWSFGQLLCDIWLSSDITCCTASILHLCVIAL
  
Inhibitor
Name:
BDBM21395
Synonyms:
3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H,3H)-quinazolinedione | 3-(2-{4-[(4-fluorophenyl)carbonyl]piperidin-1-yl}ethyl)-1,2,3,4-tetrahydroquinazoline-2,4-dione | CHEMBL1628637 | CHEMBL51 | Ketanserin | R-41,468 | R-41-468 | R41,468 | [3H]-Ketanserin
Type:
radiolabeled ligand
Emp. Form.:
C22H22FN3O3
Mol. Mass.:
395.4268
SMILES:
Fc1ccc(cc1)C(=O)C1CCN(CCn2c(=O)[nH]c3ccccc3c2=O)CC1
Structure:
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