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Target
Solute carrier family 22 member 1
Ligand
BDBM35234
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_1348
Citation
 Schwinn, DA; Johnston, GI; Page, SO; Mosley, MJ; Wilson, KH; Worman, NP; Campbell, S; Fidock, MD; Furness, LM; Parry-Smith, DJ Cloning and pharmacological characterization of human alpha-1 adrenergic receptors: sequence corrections and direct comparison with other species homologues. J Pharmacol Exp Ther 272:134-42 (1995) [PubMed] 
Target
Name:
Solute carrier family 22 member 1
Synonyms:
OCT1 | S22A1_BOVIN | SLC22A1 | adrenergic Alpha1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
62499.05
Organism:
BOVINE
Description:
adrenergic Alpha1 0 BOVINE::A7MBE0
Residue:
563
Sequence:
MLTVDDVLEQVGEFGWFQKQTFLILCLLSAAFAPIYVGIVFLAFTPDHRCRSPGVAELSRRCGWSLAEELNYTVPGPGPESQCLRYEVDWNQSTLGCLDPLASLATNGSPLPLGPCEQGWVYDTPGSSIVTEFNLVCDDSWKVDLFQSCVNLGFFLGSLGVGYIADRFGRKVCLLATTLTCASLGVLTAVAPDYTSLLIFRLLQGLVSKGSWTAGYTLITEFVGLGYRRTVAILYQMAFTVGLVLLSGLAYILPHWRWLQLAVSLPIFLLLFRFWFVPESPRWLLSQKRNTEAIKIMDHIAQKNGKLPPADLKMLSLEEDVTEKLSPSFIDLFRTPNLRKYTFILMYLWFTSSVVYQGLIMHVGATGGNLYLDFLYSALVEFPAGFIILVTIDRFGRRYPLATSNLAAGLACFLMIFIPHDLPWLNIMVACVGRMGITIVFQMVCLVNAELFPTFIRNLGMMVCSSLCDLGGVLTPFLVFRLMEVWQGSPLILFAALGLVAGGMTLLLPETKGVTLPETIEDAENLQRKAKPKENKIYLQVQTSELNTQAAERDASQGTAQQK
  
Inhibitor
Name:
BDBM35234
Synonyms:
DL-[7-3H]norepinephrine | NOREPINEPHRINE | Noradrenaline,(+) | [3H]NE
Type:
radiolabeled ligand
Emp. Form.:
C8H11NO3
Mol. Mass.:
169.1778
SMILES:
NCC(O)c1ccc(O)c(O)c1
Structure:
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