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Target
Lymphocyte antigen 96
Ligand
BDBM50239341
Substrate
n/a
Meas. Tech.
ChEMBL_1665929 (CHEMBL4015725)
IC50
5700±n/a nM
Citation
Sestito, SE; Facchini, FA; Morbioli, I; Billod, JM; Martin-Santamaria, S; Casnati, A; Sansone, F; Peri, F Amphiphilic Guanidinocalixarenes Inhibit Lipopolysaccharide (LPS)- and Lectin-Stimulated Toll-like Receptor 4 (TLR4) Signaling. J Med Chem 60:4882-4892 (2017) [PubMed] Article
More Info.:
Target
Name:
Lymphocyte antigen 96
Synonyms:
ESOP-1 | ESOP1 | ESOP1 | LY96 | LY96_HUMAN | Ly-96 | Lymphocyte antigen 96 | MD2 | Protein MD-2 | TLR4-MD2
Type:
PROTEIN
Mol. Mass.:
18551.39
Organism:
Homo sapiens (Human)
Description:
ChEMBL_107939
Residue:
160
Sequence:
MLPFLFFSTLFSSIFTEAQKQYWVCNSSDASISYTYCDKMQYPISINVNPCIELKRSKGLLHIFYIPRRDLKQLYFNLYITVNTMNLPKRKEVICRGSDDDYSFCRALKGETVNTTISFSFKGIKFSKGKYKCVVEAISGSPEEMLFCLEFVILHQPNSN