Reaction Details Report a problem with these data
Target
Advanced glycosylation end product-specific receptor
Ligand
BDBM26115
Substrate
n/a
Meas. Tech.
ChEBML_1680045
Kd
43±n/a nM
Citation
Bongarzone, S; Savickas, V; Luzi, F; Gee, AD Targeting the Receptor for Advanced Glycation Endproducts (RAGE): A Medicinal Chemistry Perspective. J Med Chem 60:7213-7232 (2017) [PubMed] Article
More Info.:
Target
Name:
Advanced glycosylation end product-specific receptor
Synonyms:
Advanced glycosylation end product-specific receptor | Ager | RAGE_RAT | Rage | Receptor for advanced glycosylation end products
Type:
PROTEIN
Mol. Mass.:
42661.10
Organism:
Rattus norvegicus
Description:
ChEMBL_105422
Residue:
402
Sequence:
MPTGTVARAWVLVLALWGAVAGGQNITARIGEPLMLSCKGAPKKPTQKLEWKLNTGRTEAWKVLSPQGDPWDSVARILPNGSLLLPAIGIVDEGTFRCRATNRLGKEVKSNYRVRVYQIPGKPEIVNPASELTANVPNKVGTCVSEGSYPAGTLSWHLDGKPLIPDGKGTVVKEETRRHPETGLFTLRSELTVTPAQGGTTPTYSCSFSLGLPRRRPLNTAPIQPRVREPLPPEGIQLLVEPEGGTVAPGGTVTLTCAISAQPPPQIHWIKDGTPLPLAPSPVLLLPEVGHEDEGIYSCVATHPSHGPQESPPVNIRVTETGDEGQAAGSVDGSGLGTLALALGILGGLGIAALLIGAILWRKRQPRLEERKAPESQEDEEERAELNQSEEAEMPENGAGGP