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Target
Solute carrier family 15 member 1
Ligand
BDBM50248190
Substrate
n/a
Meas. Tech.
ChEMBL_838489 (CHEMBL2076060)
Ki
11900000±n/a nM
Citation
 Terada, T; Saito, H; Mukai, M; Inui, K Recognition of beta-lactam antibiotics by rat peptide transporters, PEPT1 and PEPT2, in LLC-PK1 cells. Am J Physiol 273:706-11 (1997) [PubMed]  Article 
Target
Name:
Solute carrier family 15 member 1
Synonyms:
Intestinal H(+)/peptide cotransporter | Oligopeptide transporter, small intestine isoform | Pept1 | Peptide transporter 1 | Proton-coupled dipeptide cotransporter | S15A1_RAT | Slc15a1
Type:
PROTEIN
Mol. Mass.:
78933.78
Organism:
Rattus norvegicus
Description:
ChEMBL_1488841
Residue:
710
Sequence:
MGMSKSRGCFGYPLSIFFIVVNEFCERFSYYGMRALLVLYFRNFLGWDDDLSTAIYHTFVALCYLTPILGALIADSWLGKFKTIVSLSIVYTIGQAVISVSSINDLTDHDHDGSPNNLPLHVALSMIGLALIALGTGGIKPCVSAFGGDQFEEGQEKQRNRFFSIFYLAINAGSLLSTIITPILRVQQCGIHSQQACYPLAFGVPAALMAVALIVFVLGSGMYKKFQPQGNIMGKVAKCIRFAIKNRFRHRSKAFPKRNHWLDWAKEKYDERLISQIKIMTKVMFLYIPLPMFWALFDQQGSRWTLQATTMTGKIGTIEIQPDQMQTVNAILIVIMVPIVDAVVYPLIAKCGFNFTSLKKMTVGMFLASMAFVVAAIVQVEIDKTLPVFPSGNQVQIKVLNIGNNDMAVYFPGKNVTVAQMSQTDTFMTFDVDQLTSINVSSPGSPGVTTVAHEFEPGHRHTLLVWGPNLYRVVKDGLNQKPEKGENGIRFVSTLNEMITIKMSGKVYENVTSHSASNYQFFPSGQKDYTINTTEIAPNCSSDFKSSNLDFGSAYTYVIRSRASDGCLEVKEFEDIPPNTVNMALQIPQYFLLTCGEVVFSVTGLEFSYSQAPSNMKSVLQAGWLLTVAIGNIIVLIVAEAGHFDKQWAEYVLFASLLLVVCIIFAIMARFYTYINPAEIEAQFDEDEKKKGVGKENPYSSLEPVSQTNM
  
Inhibitor
Name:
BDBM50248190
Synonyms:
CHEBI:3485 | CI-983 | Cefdinir | Cefzon | FK-482 | Omnicef
Type:
Small organic molecule
Emp. Form.:
C14H13N5O5S2
Mol. Mass.:
395.414
SMILES:
[H][C@]12SCC(C=C)=C(N1C(=O)[C@H]2NC(=O)C(=N/O)\c1csc(N)n1)C(O)=O |r,c:6|
Structure:
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