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Target
Solute carrier family 15 member 1
Ligand
BDBM50485555
Substrate
n/a
Meas. Tech.
ChEMBL_838264 (CHEMBL2076212)
Ki
190000±n/a nM
Citation
 Terada, T; Sawada, K; Irie, M; Saito, H; Hashimoto, Y; Inui, K Structural requirements for determining the substrate affinity of peptide transporters PEPT1 and PEPT2. Pflugers Arch 440:679-84 (2000) [PubMed]  Article 
Target
Name:
Solute carrier family 15 member 1
Synonyms:
Intestinal H(+)/peptide cotransporter | Oligopeptide transporter, small intestine isoform | Pept1 | Peptide transporter 1 | Proton-coupled dipeptide cotransporter | S15A1_RAT | Slc15a1
Type:
PROTEIN
Mol. Mass.:
78933.78
Organism:
Rattus norvegicus
Description:
ChEMBL_1488841
Residue:
710
Sequence:
MGMSKSRGCFGYPLSIFFIVVNEFCERFSYYGMRALLVLYFRNFLGWDDDLSTAIYHTFVALCYLTPILGALIADSWLGKFKTIVSLSIVYTIGQAVISVSSINDLTDHDHDGSPNNLPLHVALSMIGLALIALGTGGIKPCVSAFGGDQFEEGQEKQRNRFFSIFYLAINAGSLLSTIITPILRVQQCGIHSQQACYPLAFGVPAALMAVALIVFVLGSGMYKKFQPQGNIMGKVAKCIRFAIKNRFRHRSKAFPKRNHWLDWAKEKYDERLISQIKIMTKVMFLYIPLPMFWALFDQQGSRWTLQATTMTGKIGTIEIQPDQMQTVNAILIVIMVPIVDAVVYPLIAKCGFNFTSLKKMTVGMFLASMAFVVAAIVQVEIDKTLPVFPSGNQVQIKVLNIGNNDMAVYFPGKNVTVAQMSQTDTFMTFDVDQLTSINVSSPGSPGVTTVAHEFEPGHRHTLLVWGPNLYRVVKDGLNQKPEKGENGIRFVSTLNEMITIKMSGKVYENVTSHSASNYQFFPSGQKDYTINTTEIAPNCSSDFKSSNLDFGSAYTYVIRSRASDGCLEVKEFEDIPPNTVNMALQIPQYFLLTCGEVVFSVTGLEFSYSQAPSNMKSVLQAGWLLTVAIGNIIVLIVAEAGHFDKQWAEYVLFASLLLVVCIIFAIMARFYTYINPAEIEAQFDEDEKKKGVGKENPYSSLEPVSQTNM
  
Inhibitor
Name:
BDBM50485555
Synonyms:
CHEMBL55636 | Gly-Leu-Tyr
Type:
Small organic molecule
Emp. Form.:
C17H25N3O5
Mol. Mass.:
351.3975
SMILES:
CC(C)C[C@H](NC(=O)CN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(O)=O
Structure:
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