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Target
Solute carrier family 15 member 1
Ligand
BDBM50485607
Substrate
n/a
Meas. Tech.
ChEMBL_836467 (CHEMBL2076907)
Ki
3600000±n/a nM
Citation
 Sawada, K; Terada, T; Saito, H; Hashimoto, Y; Inui, KI Recognition of L-amino acid ester compounds by rat peptide transporters PEPT1 and PEPT2. J Pharmacol Exp Ther 291:705-9 (1999) [PubMed] 
Target
Name:
Solute carrier family 15 member 1
Synonyms:
Intestinal H(+)/peptide cotransporter | Oligopeptide transporter, small intestine isoform | Pept1 | Peptide transporter 1 | Proton-coupled dipeptide cotransporter | S15A1_RAT | Slc15a1
Type:
PROTEIN
Mol. Mass.:
78933.78
Organism:
Rattus norvegicus
Description:
ChEMBL_1488841
Residue:
710
Sequence:
MGMSKSRGCFGYPLSIFFIVVNEFCERFSYYGMRALLVLYFRNFLGWDDDLSTAIYHTFVALCYLTPILGALIADSWLGKFKTIVSLSIVYTIGQAVISVSSINDLTDHDHDGSPNNLPLHVALSMIGLALIALGTGGIKPCVSAFGGDQFEEGQEKQRNRFFSIFYLAINAGSLLSTIITPILRVQQCGIHSQQACYPLAFGVPAALMAVALIVFVLGSGMYKKFQPQGNIMGKVAKCIRFAIKNRFRHRSKAFPKRNHWLDWAKEKYDERLISQIKIMTKVMFLYIPLPMFWALFDQQGSRWTLQATTMTGKIGTIEIQPDQMQTVNAILIVIMVPIVDAVVYPLIAKCGFNFTSLKKMTVGMFLASMAFVVAAIVQVEIDKTLPVFPSGNQVQIKVLNIGNNDMAVYFPGKNVTVAQMSQTDTFMTFDVDQLTSINVSSPGSPGVTTVAHEFEPGHRHTLLVWGPNLYRVVKDGLNQKPEKGENGIRFVSTLNEMITIKMSGKVYENVTSHSASNYQFFPSGQKDYTINTTEIAPNCSSDFKSSNLDFGSAYTYVIRSRASDGCLEVKEFEDIPPNTVNMALQIPQYFLLTCGEVVFSVTGLEFSYSQAPSNMKSVLQAGWLLTVAIGNIIVLIVAEAGHFDKQWAEYVLFASLLLVVCIIFAIMARFYTYINPAEIEAQFDEDEKKKGVGKENPYSSLEPVSQTNM
  
Inhibitor
Name:
BDBM50485607
Synonyms:
CHEMBL1209949 | L-Valine Methyl Ester
Type:
Small organic molecule
Emp. Form.:
C6H13NO2
Mol. Mass.:
131.1729
SMILES:
COC(=O)[C@@H](N)C(C)C |r|
Structure:
Search PDB for entries with ligand similarity: