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Target
PHD finger protein 23
Ligand
BDBM50440571
Substrate
n/a
Meas. Tech.
ChEMBL_1300213 (CHEMBL3136677)
IC50
>30000±n/a nM
Citation
 Camerino, MA; Zhong, N; Dong, A; Dickson, BM; James, LI; Baughman, BM; Norris, JL; Kireev, DB; Janzen, WP; Arrowsmith, CH; Frye, SV The structure-activity relationships of L3MBTL3 inhibitors: flexibility of the dimer interface. Medchemcomm 4:1501-1507 (2013) [PubMed]  Article 
Target
Name:
PHD finger protein 23
Synonyms:
PDH-containing protein JUNE-1 | PHD finger protein 23 | PHD finger protein 23 (PHF23) | PHF23 | PHF23_HUMAN
Type:
Protein
Mol. Mass.:
43813.67
Organism:
Homo sapiens (Human)
Description:
n/a
Residue:
403
Sequence:
MLEAMAEPSPEDPPPTLKPETQPPEKRRRTIEDFNKFCSFVLAYAGYIPPSKEESDWPASGSSSPLRGESAADSDGWDSAPSDLRTIQTFVKKAKSSKRRAAQAGPTQPGPPRSTFSRLQAPDSATLLEKMKLKDSLFDLDGPKVASPLSPTSLTHTSRPPAALTPVPLSQGDLSHPPRKKDRKNRKLGPGAGAGFGVLRRPRPTPGDGEKRSRIKKSKKRKLKKAERGDRLPPPGPPQAPPSDTDSEEEEEEEEEEEEEEMATVVGGEAPVPVLPTPPEAPRPPATVHPEGVPPADSESKEVGSTETSQDGDASSSEGEMRVMDEDIMVESGDDSWDLITCYCRKPFAGRPMIECSLCGTWIHLSCAKIKKTNVPDFFYCQKCKELRPEARRLGGPPKSGEP
  
Inhibitor
Name:
BDBM50440571
Synonyms:
CHEMBL2426474
Type:
Small organic molecule
Emp. Form.:
C28H42N4O2
Mol. Mass.:
466.6587
SMILES:
O=C(N1CCC(CC1)N1CCCCC1)c1ccc(cc1)C(=O)N1CCC(CC1)N1CCCCC1
Structure:
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