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Target
Transmembrane domain-containing protein TMIGD3
Ligand
BDBM50500485
Substrate
n/a
Meas. Tech.
ChEMBL_1543585 (CHEMBL3750703)
Kd
741±n/a nM
Citation
 Ranganathan, A; Stoddart, LA; Hill, SJ; Carlsson, J Fragment-Based Discovery of Subtype-Selective Adenosine Receptor Ligands from Homology Models. J Med Chem 58:9578-90 (2015) [PubMed]  Article 
Target
Name:
Transmembrane domain-containing protein TMIGD3
Synonyms:
TMIG3_HUMAN | TMIGD3 | Transmembrane domain-containing protein TMIGD3
Type:
PROTEIN
Mol. Mass.:
30335.79
Organism:
Homo sapiens (Human)
Description:
ChEMBL_114868
Residue:
266
Sequence:
MEGSPAGPIEQKEARWESSWEEQPDWTLGCLSPESQFRIPGLPGCILSFQLKVCFLPVMWLFILLSLALISDAMVMDEKVKRSFVLDTASAICNYNAHYKNHPKYWCRGYFRDYCNIIAFSPNSTNHVALRDTGNQLIVTMSCLTKEDTGWYWCGIQRDFARDDMDFTELIVTDDKGTLANDFWSGKDLSGNKTRSCKAPKVVRKADRSRTSILIICILITGLGIISVISHLTKRRRSQRNRRVGNTLKPFSRVLTPKEMAPTEQM
  
Inhibitor
Name:
BDBM50500485
Synonyms:
CHEMBL3745803
Type:
Small organic molecule
Emp. Form.:
C12H10N2O2S
Mol. Mass.:
246.285
SMILES:
CCc1cc2c(nc([nH]c2=O)-c2ccoc2)s1
Structure:
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