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Target
Xaa-Pro dipeptidase
Ligand
BDBM50240386
Substrate
n/a
Meas. Tech.
ChEBML_159886
Ki
960000±n/a nM
Citation
 Kumaravel, G; Boettcher, BR; Shapiro, MJ; Petter, C Peptide mimics of glycylproline as inhibitors of prolidase Bioorg Med Chem Lett 5:2825-2828 (1995)    Article 
Target
Name:
Xaa-Pro dipeptidase
Synonyms:
PEPD | PEPD_HUMAN | PRD
Type:
PROTEIN
Mol. Mass.:
54541.05
Organism:
Homo sapiens (Human)
Description:
ChEMBL_159887
Residue:
493
Sequence:
MAAATGPSFWLGNETLKVPLALFALNRQRLCERLRKNPAVQAGSIVVLQGGEETQRYCTDTGVLFRQESFFHWAFGVTEPGCYGVIDVDTGKSTLFVPRLPASHATWMGKIHSKEHFKEKYAVDDVQYVDEIASVLTSQKPSVLLTLRGVNTDSGSVCREASFDGISKFEVNNTILHPEIVECRVFKTDMELEVLRYTNKISSEAHREVMKAVKVGMKEYELESLFEHYCYSRGGMRHSSYTCICGSGENSAVLHYGHAGAPNDRTIQNGDMCLFDMGGEYYCFASDITCSFPANGKFTADQKAVYEAVLRSSRAVMGAMKPGVWWPDMHRLADRIHLEELAHMGILSGSVDAMVQAHLGAVFMPHGLGHFLGIDVHDVGGYPEGVERIDEPGLRSLRTARHLQPGMVLTVEPGIYFIDHLLDEALADPARASFLNREVLQRFRGFGGVRIEEDVVVTDSGIELLTCVPRTVEEIEACMAGCDKAFTPFSGPK
  
Inhibitor
Name:
BDBM50240386
Synonyms:
5-amino-4-oxopentanoic acid | 5-aminolevulinic acid | AMINOLEVULINIC ACID | Aminolevulinic Acid Hydrochloride | CHEMBL601 | Levulan | delta-aminolevulinic acid
Type:
Small organic molecule
Emp. Form.:
C5H9NO3
Mol. Mass.:
131.1299
SMILES:
NCC(=O)CCC(O)=O
Structure:
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