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Target
VIM-1 protein
Ligand
BDBM26116
Substrate
n/a
Meas. Tech.
ChEMBL_678224 (CHEMBL1280219)
IC50
41600±n/a nM
Citation
 Juan, C; Beceiro, A; Gutiérrez, O; Albertí, S; Garau, M; Pérez, JL; Bou, G; Oliver, A Characterization of the new metallo-beta-lactamase VIM-13 and its integron-borne gene from a Pseudomonas aeruginosa clinical isolate in Spain. Antimicrob Agents Chemother 52:3589-96 (2008) [PubMed]  Article 
Target
Name:
VIM-1 protein
Synonyms:
Beta-lactamase VIM-1 | Class B carbapenemase VIM-1 | Metallo-beta-lactamase VIM-1 | Metallobeta-lactamase | VIM-1 | VIM-1 metallo-beta lactamase | VIM-1 metallo-beta-lactamase | VIM-1 protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28014.53
Organism:
Pseudomonas aeruginosa
Description:
n/a
Residue:
266
Sequence:
MLKVISSLLVYMTASVMAVASPLAHSGEPSGEYPTVNEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEAEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSANVLYGGCAVHELSSTSAGNVADADLAEWPTSVERIQKHYPEAEVVIPGHGLPGGLDLLQHTANVVKAHKNRSVAE
  
Inhibitor
Name:
BDBM26116
Synonyms:
CHEMBL284104 | Dipicolinate | pyridine carboxylate, 6d | pyridine-2,6-dicarboxylic acid
Type:
Small organic molecule
Emp. Form.:
C7H5NO4
Mol. Mass.:
167.1189
SMILES:
OC(=O)c1cccc(n1)C(O)=O
Structure:
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