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Target
Muscarinic receptor M1
Ligand
BDBM50055978
Substrate
n/a
Meas. Tech.
ChEMBL_140161 (CHEMBL745466)
Ki
0.02±n/a nM
Citation
 Visser, TJ; van Waarde, A; Jansen, TJ; Visser, GM; van der Mark, TW; Kraan, J; Ensing, K; Vaalburg, W Stereoselective synthesis and biodistribution of potent [11C]-labeled antagonists for positron emission tomography imaging of muscarinic receptors in the airways. J Med Chem 40:117-24 (1997) [PubMed]  Article 
Target
Name:
Muscarinic receptor M1
Synonyms:
Muscarinic acetylcholine receptor M1
Type:
PROTEIN
Mol. Mass.:
15022.43
Organism:
Bos taurus
Description:
ChEMBL_140161
Residue:
139
Sequence:
ETENRARELAALQGSETPGKGGGSSSSSERSQPGAEGSPETPPGRCCRCCRTPRLLQAYSWKEEEEEDEGSMESLTSSEGEEPGSEVVIKMPMVDPEAQAPAKQPPRSSPNTVKRPTRKGRERAGKGQKPRGKEQLAKR
  
Inhibitor
Name:
BDBM50055978
Synonyms:
4-((R)-2-Cyclohexyl-2-hydroxy-2-phenyl-acetoxy)-1,1-dimethyl-piperidinium; iodide | CHEMBL21905
Type:
Small organic molecule
Emp. Form.:
C21H32NO3
Mol. Mass.:
346.4831
SMILES:
C[N+]1(C)CCC(CC1)OC(=O)[C@@](O)(C1CCCCC1)c1ccccc1
Structure:
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