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Target
RuvB-like 1
Ligand
BDBM50015300
Substrate
n/a
Meas. Tech.
ChEMBL_1349809 (CHEMBL3268010)
IC50
18000±n/a nM
Citation
Elkaim, J; Lamblin, M; Laguerre, M; Rosenbaum, J; Lestienne, P; Eloy, L; Cresteil, T; Felpin, FX; Dessolin, J Design, synthesis and biological evaluation of Pontin ATPase inhibitors through a molecular docking approach. Bioorg Med Chem Lett 24:2512-6 (2014) [PubMed] Article
More Info.:
Target
Name:
RuvB-like 1
Synonyms:
49 kDa TATA box-binding protein-interacting protein | 49 kDa TBP-interacting protein | 54 kDa erythrocyte cytosolic protein | ECP-54 | INO80 complex subunit H | INO80H | NMP 238 | NMP238 | Nuclear matrix protein 238 | Pontin 52 | RUVB1_HUMAN | RUVBL1 | TAP54-alpha | TIP49 | TIP49A | TIP60-associated protein 54-alpha
Type:
PROTEIN
Mol. Mass.:
50226.43
Organism:
Homo sapiens (Human)
Description:
ChEMBL_108308
Residue:
456
Sequence:
MKIEEVKSTTKTQRIASHSHVKGLGLDESGLAKQAASGLVGQENAREACGVIVELIKSKKMAGRAVLLAGPPGTGKTALALAIAQELGSKVPFCPMVGSEVYSTEIKKTEVLMENFRRAIGLRIKETKEVYEGEVTELTPCETENPMGGYGKTISHVIIGLKTAKGTKQLKLDPSIFESLQKERVEAGDVIYIEANSGAVKRQGRCDTYATEFDLEAEEYVPLPKGDVHKKKEIIQDVTLHDLDVANARPQGGQDILSMMGQLMKPKKTEITDKLRGEINKVVNKYIDQGIAELVPGVLFVDEVHMLDIECFTYLHRALESSIAPIVIFASNRGNCVIRGTEDITSPHGIPLDLLDRVMIIRTMLYTPQEMKQIIKIRAQTEGINISEEALNHLGEIGTKTTLRYSVQLLTPANLLAKINGKDSIEKEHVEEISELFYDAKSSAKILADQQDKYMK