Reaction Details Report a problem with these data
Target
Similar to alpha-tubulin isoform 1
Ligand
BDBM50035218
Substrate
n/a
Meas. Tech.
ChEMBL_1457783 (CHEMBL3369800)
IC50
830±n/a nM
Citation
Kamal, A; Srinivasa Reddy, T; Polepalli, S; Shalini, N; Reddy, VG; Subba Rao, AV; Jain, N; Shankaraiah, N Synthesis and biological evaluation of podophyllotoxin congeners as tubulin polymerization inhibitors. Bioorg Med Chem 22:5466-75 (2014) [PubMed] Article
More Info.:
Target
Name:
Similar to alpha-tubulin isoform 1
Synonyms:
Similar to alpha-tubulin isoform 1
Type:
PROTEIN
Mol. Mass.:
10383.05
Organism:
Bos taurus
Description:
ChEMBL_104716
Residue:
99
Sequence:
CVSASPSTLARLVSRSAMPAGSSTAWNTAFSPMARCQVTKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRSSSTLSSSSQAKKMP