Reaction Details Report a problem with these data
Target
Adiponectin receptor protein 1
Ligand
BDBM50059083
Substrate
n/a
Meas. Tech.
ChEMBL_1461017 (CHEMBL3395075)
Kd
1800±n/a nM
Citation
Rana, S; Blowers, EC; Natarajan, A Small molecule adenosine 5'-monophosphate activated protein kinase (AMPK) modulators and human diseases. J Med Chem 58:2-29 (2015) [PubMed] Article
More Info.:
Target
Name:
Adiponectin receptor protein 1
Synonyms:
ADIPOR1 | Adiponectin receptor protein 1 | PAQR1 | PAQR1 | PAQR1_HUMAN | Progestin and adipoQ receptor family member I | TESBP1A
Type:
PROTEIN
Mol. Mass.:
42619.21
Organism:
Homo sapiens (Human)
Description:
ChEMBL_109558
Residue:
375
Sequence:
MSSHKGSVVAQGNGAPASNREADTVELAELGPLLEEKGKRVIANPPKAEEEQTCPVPQEEEEEVRVLTLPLQAHHAMEKMEEFVYKVWEGRWRVIPYDVLPDWLKDNDYLLHGHRPPMPSFRACFKSIFRIHTETGNIWTHLLGFVLFLFLGILTMLRPNMYFMAPLQEKVVFGMFFLGAVLCLSFSWLFHTVYCHSEKVSRTFSKLDYSGIALLIMGSFVPWLYYSFYCSPQPRLIYLSIVCVLGISAIIVAQWDRFATPKHRQTRAGVFLGLGLSGVVPTMHFTIAEGFVKATTVGQMGWFFLMAVMYITGAGLYAARIPERFFPGKFDIWFQSHQIFHVLVVAAAFVHFYGVSNLQEFRYGLEGGCTDDTLL