Reaction Details Report a problem with these data
Target
Nucleophosmin
Ligand
BDBM50094238
Substrate
n/a
Meas. Tech.
ChEMBL_1502715 (CHEMBL3590711)
EC50
2500±n/a nM
Citation
Penthala, NR; Crooks, PA; Freeman, ML; Sekhar, KR Development and validation of a novel assay to identify radiosensitizers that target nucleophosmin 1. Bioorg Med Chem 23:3681-6 (2015) [PubMed] Article
More Info.:
Target
Name:
Nucleophosmin
Synonyms:
NPM | NPM/ALK (Nucleophosmin/ALK tyrosine kinase receptor) | NPM1 | NPM_HUMAN
Type:
PROTEIN
Mol. Mass.:
32552.99
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1502715
Residue:
294
Sequence:
MEDSMDMDMSPLRPQNYLFGCELKADKDYHFKVDNDENEHQLSLRTVSLGAGAKDELHIVEAEAMNYEGSPIKVTLATLKMSVQPTVSLGGFEITPPVVLRLKCGSGPVHISGQHLVAVEEDAESEDEEEEDVKLLSISGKRSAPGGGSKVPQKKVKLAADEDDDDDDEEDDDEDDDDDDFDDEEAEEKAPVKKSIRDTPAKNAQKSNQNGKDSKPSSTPRSKGQESFKKQEKTPKTPKGPSSVEDIKAKMQASIEKGGSLPKVEAKFINYVKNCFRMTDQEAIQDLWQWRKSL