Reaction Details Report a problem with these data
Target
Adenosine receptor A1
Ligand
BDBM82557
Substrate
n/a
Ki
4±n/a nM
Comments
PDSP_945
Citation
Hill, RJ; Oleynek, JJ; Hoth, CF; Kiron, MA; Weng, W; Wester, RT; Tracey, WR; Knight, DR; Buchholz, RA; Kennedy, SP Cloning, expression and pharmacological characterization of rabbit adenosine A1 and A3 receptors. J Pharmacol Exp Ther 280:122-8 (1997) [PubMed]
More Info.:
Target
Name:
Adenosine receptor A1
Synonyms:
AA1R_RABIT | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | ADORA1 | Adenosine receptor A1 (A1)
Type:
Enzyme
Mol. Mass.:
36566.33
Organism:
Oryctolagus cuniculus (Rabbit)
Description:
P34970
Residue:
328
Sequence:
MPPSISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGALVIPLAILINIGPETYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKAVVTPRRAAVAIAGCWILSLVVGLTPMFGWNNLREVQRAWAANGSVGEPVIKCEFEKVISMEYMVYFNFFVWVLPPLLLMVLIYLEVFYLIRRQLSKKASASSGDPHKYYGKELKIAKSLALILFLFALSWLPLHILNCVTLFCPSCQKPSILVYTAIFLTHGNSAMNPIVYAFRIHKFRVTFLKIWNDHFRCRPAPAGDGDEDLPEEKPND