Reaction Details Report a problem with these data
Target
Muscarinic acetylcholine receptor M4
Ligand
BDBM82371
Substrate
n/a
Ki
57.54±n/a nM
Comments
PDSP_1918
Citation
Chelala, JL; Kilani, A; Miller, MJ; Martin, RJ; Ernsberger, P Muscarinic receptor binding sites of the M4 subtype in porcine lung parenchyma. Pharmacol Toxicol 83:200-7 (1998) [PubMed] Article
More Info.:
Target
Name:
Muscarinic acetylcholine receptor M4
Synonyms:
CHRM4 | CHRM4 protein | Cholinergic, muscarinic M4
Type:
Enzyme Catalytic Domain
Mol. Mass.:
30028.84
Organism:
bovine
Description:
A6QQE4
Residue:
271
Sequence:
MTVLYVHISLASRSRVHKHRPEGPKEKKAKTLAFLKSPLMKQSVKKPPPPGDTTARGELRNGKLEEAPPPVLPPPPRPMADKDTSNESSSGSATQNTKERPPTELSTTEATTPATPAPPLQPRTLNPASKWSKIQIVTKQTGNECVTAIEIVPATPAGMRPAANVARKFASIARSQVRKKRQMAARERKVTRTIFAILLAFILTWTPYNVMVLVNTFCQSCIPETVWSIGYWLCYVNSTINPACYALCNATFKKTFRHLLLCQYRNIGTAR