Reaction Details
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Report a problem with these dataTarget
Adenosine receptor A3
Ligand
BDBM85036
Substrate
n/a
Ki
36.6±n/a nM
Comments
PDSP_458
Citation
Durand, IH; Green, RD Cloning of a chick A3 adenosine receptor: characterization of ligand binding and receptor-effector coupling of chick A1 and A3 adenosine receptors. Naunyn Schmiedebergs Arch Pharmacol 363:81-6 (2001) [PubMed] Article More Info.:
Target
Name:
Adenosine receptor A3
Synonyms:
ADENOSINE A3 | ADORA3
Type:
Enzyme Catalytic Domain
Mol. Mass.:
37723.59
Organism:
Chick
Description:
A0A8V1ACC1
Residue:
338
Sequence:
MCPQGSPCPASSSPINVTFNTSQVMGSIDVIYISAECLVALLAALGNIPVVWAVKLNAAFHNTTMYFIASLALADIAVGVFVVPLAVLVSLQVSIPFHFCLFLCCLMVVFTQASILSLLAIAIDRYLRVKLPIRYKIISTERRIWGALGLCWSLSLLVGLTPMFGWNKQRSAPYHTCGFTSVIRMDYMVYFSFFAWTLIPLSIMCALYVAVFYIIRTKLSQGATGARGAGTFYGKEFRKAKSLALILFLFAVSWLPLCIMNCVLYFHPEYKIPKPWIFLGILLSHANSAMNPVVYACKIKKFKTTYLLILRTYILCRKKPQAMPSSYRLNTPAVVDTE
Inhibitor
Name:
BDBM85036
Synonyms:
BW-A1433 | BWA1433 | CAS_129447 | NSC_129447
Type:
Small organic molecule
Emp. Form.:
C20H22N4O4
Mol. Mass.:
382.4131
SMILES:
CCCn1c2nc([nH]c2c(=O)n(CCC)c1=O)-c1ccc(C=CC(O)=O)cc1 |w:21.22|
Structure:
