Reaction Details Report a problem with these data
Target
Histamine H1 receptor
Ligand
BDBM86748
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_7576
Citation
Deecher, DC; Beyer, CE; Johnston, G; Bray, J; Shah, S; Abou-Gharbia, M; Andree, TH Desvenlafaxine succinate: A new serotonin and norepinephrine reuptake inhibitor. J Pharmacol Exp Ther 318:657-65 (2006) [PubMed] Article
More Info.:
Target
Name:
Histamine H1 receptor
Synonyms:
HISTAMINE H1 | HRH1 | HRH1 protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
56008.28
Organism:
BOVINE
Description:
A5D795
Residue:
491
Sequence:
MTCPNSSCVFEDKMCEGNKTAPANNAQLTPLVVVLSTISLVTVGLNLLVLYAVRSERKLHTVGNLYIVSLSVADLIVGVVVMPMNILYLLMSRWSLGRPLCLFWLSMDYVASTASIFSVFILCIDRYRSVQQPLKYLRYRTKTRASITILAAWFLSFLWIIPILGWRHFQPKTPEPREDKCETDFYNVTWFKVMTAIINFYLPTLLMLWFYAKIYKAVRQHCQHRELINGSFPSFSDMKMKPENLQVGTKKPGKESPWEVLKRKPKDTGGGPVLKPPSQEPKEVTSPGVFSQEKEEKDGELGKYYCFPLDTVQAQPEAEGSGRGYAAINQSQNQLEMGEQGLSMPGAKEALEDQILGDSQSFSRTDSDTPAEPALAKGKSRSESSTGLEYIKFTWKRLRSHSRQYVSGLHMNRERKAAKQLGFIMAAFIICWIPYFIFFMVIAFCESCCNQHVHMFTIWLGYINSTLNPLIYPLCNENFKKTFKKILHIRS