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Target
Melanocortin receptor 4
Ligand
BDBM43425
Substrate
n/a
Meas. Tech.
Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R)
EC50
>89263±n/a nM
Citation
 PubChem, PC Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM43425
Synonyms:
MLS000392773 | N-[(2-chlorophenyl)methylideneamino]-2-benzo[cd]indolamine | N-[(2-chlorophenyl)methylideneamino]benzo[cd]indol-2-amine | SMR000261714 | benzo[cd]indol-2-yl-[(2-chlorobenzylidene)amino]amine | benzo[cd]indol-2-yl-[(E)-(2-chlorobenzylidene)amino]amine | cid_2315072
Type:
Small organic molecule
Emp. Form.:
C18H12ClN3
Mol. Mass.:
305.761
SMILES:
Clc1ccccc1C=NNC1=Nc2cccc3cccc1c23 |w:8.9,t:11|
Structure:
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