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Target
Melanocortin receptor 4
Ligand
BDBM50563
Substrate
n/a
Meas. Tech.
Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R)
EC50
>89178±n/a nM
Citation
 PubChem, PC Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM50563
Synonyms:
4-[4-(6-phenyl-4-thieno[2,3-d]pyrimidinyl)-1-piperazinyl]phenol | 4-[4-(6-phenylthieno[2,3-d]pyrimidin-4-yl)piperazin-1-yl]phenol | 4-[4-(6-phenylthieno[2,3-d]pyrimidin-4-yl)piperazino]phenol | MLS000760381 | SMR000369638 | cid_2495129
Type:
Small organic molecule
Emp. Form.:
C22H20N4OS
Mol. Mass.:
388.485
SMILES:
Oc1ccc(cc1)N1CCN(CC1)c1ncnc2sc(cc12)-c1ccccc1
Structure:
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