Target
Melanocortin receptor 4
Ligand
BDBM78963
Substrate
n/a
Meas. Tech.
Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R)
EC50
>89131±n/a nM
Citation
 PubChem, PC Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM78963
Synonyms:
MLS001205948 | N-(4,5-Dihydro-1H-imidazol-2-yl)-N'-[1-(4-hexyloxy-phenyl)-ethylidene]-hydrazine | N-[1-(4-hexoxyphenyl)ethylideneamino]-4,5-dihydro-1H-imidazol-2-amine | SMR000513357 | [(E)-1-(4-hexoxyphenyl)ethylideneamino]-(2-imidazolin-2-yl)amine | [1-(4-hexoxyphenyl)ethylideneamino]-(2-imidazolin-2-yl)amine | cid_3098371
Type:
Small organic molecule
Emp. Form.:
C17H26N4O
Mol. Mass.:
302.4145
SMILES:
CCCCCCOc1ccc(cc1)C(C)=NNC1=NCCN1 |w:15.16,t:18|
Structure:
Search PDB for entries with ligand similarity: