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Target
Melanocortin receptor 4
Ligand
BDBM48733
Substrate
n/a
Meas. Tech.
Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R)
EC50
>89228±n/a nM
Citation
 PubChem, PC Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM48733
Synonyms:
1-cetyl-N,N-diethyl-pyridin-1-ium-3-carboxamide;bromide | 1-cetyl-N,N-diethyl-pyridin-1-ium-3-carboxamide;chloride | 3-Diethylcarbamoyl-1-hexadecyl-pyridinium | MLS000587364 | N,N-diethyl-1-hexadecyl-3-pyridin-1-iumcarboxamide;bromide | N,N-diethyl-1-hexadecyl-pyridin-1-ium-3-carboxamide;bromide | N,N-diethyl-1-hexadecylpyridin-1-ium-3-carboxamide;bromide | SMR000211414 | cid_12005597
Type:
Small organic molecule
Emp. Form.:
C26H47N2O
Mol. Mass.:
403.6636
SMILES:
CCCCCCCCCCCCCCCC[n+]1cccc(c1)C(=O)N(CC)CC
Structure:
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