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Target
Melanocortin receptor 4
Ligand
BDBM88513
Substrate
n/a
Meas. Tech.
Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R)
EC50
>89224±n/a nM
Citation
 PubChem, PC Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM88513
Synonyms:
MLS003124204 | N-[3,6-bis(3,4-dimethoxyphenyl)-8-imidazo[1,2-a]pyridinyl]acetamide | N-[3,6-bis(3,4-dimethoxyphenyl)imidazo[1,2-a]pyridin-8-yl]acetamide | N-[3,6-bis(3,4-dimethoxyphenyl)imidazo[1,2-a]pyridin-8-yl]ethanamide | SMR001292710 | cid_46943460
Type:
Small organic molecule
Emp. Form.:
C25H25N3O5
Mol. Mass.:
447.4831
SMILES:
COc1ccc(cc1OC)-c1cnc2c(NC(C)=O)cc(cn12)-c1ccc(OC)c(OC)c1
Structure:
Search PDB for entries with ligand similarity: