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Target
Melanocortin receptor 4
Ligand
BDBM40530
Substrate
n/a
Meas. Tech.
TRFRET-based cell-based high throughput dose response assay for biased ligands (antagonists) of the melanocortin 4 receptor (MC4R)
IC50
>64598±n/a nM
Citation
 PubChem, PC TRFRET-based cell-based high throughput dose response assay for biased ligands (antagonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM40530
Synonyms:
4-chloranyl-8-(diethylamino)pyrano[3,2-c]chromene-2,5-dione | 4-chloro-8-(diethylamino)-2H,5H-pyrano[3,2-c]chromene-2,5-dione | 4-chloro-8-(diethylamino)pyrano[3,2-c][1]benzopyran-2,5-dione | 4-chloro-8-(diethylamino)pyrano[3,2-c]chromene-2,5-dione | 4-chloro-8-(diethylamino)pyrano[3,2-c]chromene-2,5-quinone | MLS000059194 | SMR000069566 | cid_756377
Type:
Small organic molecule
Emp. Form.:
C16H14ClNO4
Mol. Mass.:
319.74
SMILES:
CCN(CC)c1ccc2c(c1)oc(=O)c1c(Cl)cc(=O)oc21
Structure:
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