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Target
Melanocortin receptor 4
Ligand
BDBM88594
Substrate
n/a
Meas. Tech.
TRFRET-based cell-based high throughput dose response assay for biased ligands (antagonists) of the melanocortin 4 receptor (MC4R)
IC50
>64579±n/a nM
Citation
 PubChem, PC TRFRET-based cell-based high throughput dose response assay for biased ligands (antagonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM88594
Synonyms:
2-(4-ethylphenoxy)-N-[2,2,2-trichloro-1-({[(2-methoxyphenyl)amino]carbonothioyl}amino)ethyl]acetamide | 2-(4-ethylphenoxy)-N-[2,2,2-trichloro-1-[(2-methoxyphenyl)carbamothioylamino]ethyl]acetamide | 2-(4-ethylphenoxy)-N-[2,2,2-trichloro-1-[(2-methoxyphenyl)thiocarbamoylamino]ethyl]acetamide | 2-(4-ethylphenoxy)-N-[2,2,2-trichloro-1-[[(2-methoxyanilino)-sulfanylidenemethyl]amino]ethyl]acetamide | 2-(4-ethylphenoxy)-N-[2,2,2-tris(chloranyl)-1-[(2-methoxyphenyl)carbamothioylamino]ethyl]ethanamide | MLS000573507 | SMR000195010 | cid_2898120
Type:
Small organic molecule
Emp. Form.:
C20H22Cl3N3O3S
Mol. Mass.:
490.831
SMILES:
CCc1ccc(OCC(=O)NC(NC(=S)Nc2ccccc2OC)C(Cl)(Cl)Cl)cc1
Structure:
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