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Target
Melanocortin receptor 4
Ligand
BDBM88633
Substrate
n/a
Meas. Tech.
TRFRET-based cell-based high throughput dose response assay for biased ligands (antagonists) of the melanocortin 4 receptor (MC4R)
IC50
>64586±n/a nM
Citation
 PubChem, PC TRFRET-based cell-based high throughput dose response assay for biased ligands (antagonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM88633
Synonyms:
4-chloranyl-3-nitro-N-(2-piperidin-1-ylphenyl)benzamide | 4-chloro-3-nitro-N-(2-piperidin-1-ylphenyl)benzamide | 4-chloro-3-nitro-N-(2-piperidinophenyl)benzamide | 4-chloro-3-nitro-N-[2-(1-piperidinyl)phenyl]benzamide | MLS000517347 | SMR000343460 | cid_2161746
Type:
Small organic molecule
Emp. Form.:
C18H18ClN3O3
Mol. Mass.:
359.807
SMILES:
[O-][N+](=O)c1cc(ccc1Cl)C(=O)Nc1ccccc1N1CCCCC1
Structure:
Search PDB for entries with ligand similarity: