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Target
Melanocortin receptor 4
Ligand
BDBM71167
Substrate
n/a
Meas. Tech.
TRFRET-based cell-based high throughput dose response assay for biased ligands (antagonists) of the melanocortin 4 receptor (MC4R)
IC50
>64542±n/a nM
Citation
 PubChem, PC TRFRET-based cell-based high throughput dose response assay for biased ligands (antagonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM71167
Synonyms:
2-chloranyl-N-(4-chlorophenyl)-N-(1-ethanoylindol-3-yl)ethanamide | MLS000333023 | N-(1-Acetyl-1H-indol-3-yl)-2-chloro-N-(4-chloro-phenyl)-acetamide | N-(1-acetyl-3-indolyl)-2-chloro-N-(4-chlorophenyl)acetamide | N-(1-acetylindol-3-yl)-2-chloro-N-(4-chlorophenyl)acetamide | SMR000436335 | cid_2017227
Type:
Small organic molecule
Emp. Form.:
C18H14Cl2N2O2
Mol. Mass.:
361.222
SMILES:
CC(=O)n1cc(N(C(=O)CCl)c2ccc(Cl)cc2)c2ccccc12
Structure:
Search PDB for entries with ligand similarity: