Reaction Details Report a problem with these data
Target
V-type proton ATPase subunit c'
Ligand
BDBM3699
Substrate
n/a
Meas. Tech.
Dose Response with BCECF Assay for V-ATPase inhibitors that increase vacuolar pH, Powder Set 1
EC50
860±n/a nM
Citation
 PubChem, PC Dose Response with BCECF Assay for V-ATPase inhibitors that increase vacuolar pH, Powder Set 1 PubChem Bioassay (2012)[AID] 
Target
Name:
V-type proton ATPase subunit c'
Synonyms:
CLS9 | TFP3 | VATL2_YEAST | VMA11 | Vma11p
Type:
Enzyme Catalytic Domain
Mol. Mass.:
17039.28
Organism:
Saccharomyces cerevisiae S288c
Description:
gi_6325022
Residue:
164
Sequence:
MSTQLASNIYAPLYAPFFGFAGCAAAMVLSCLGAAIGTAKSGIGIAGIGTFKPELIMKSLIPVVMSGILAIYGLVVAVLIAGNLSPTEDYTLFNGFMHLSCGLCVGFACLSSGYAIGMVGDVGVRKYMHQPRLFVGIVLILIFSEVLGLYGMIVALILNTRGSE
  
Inhibitor
Name:
BDBM3699
Synonyms:
cid_7292627
Type:
n/a
Emp. Form.:
C16H13ClN4O4S
Mol. Mass.:
392.817
SMILES:
[O-][N+](=O)c1ccc(o1)C(=O)N1CCN(CC1)c1nc2c(Cl)cccc2s1
Structure:
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