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Target
V-type proton ATPase subunit c'
Ligand
BDBM3738
Substrate
n/a
Meas. Tech.
Dose Response with BCECF Assay for V-ATPase inhibitors that increase vacuolar pH, Powder Set 1
EC50
1588±n/a nM
Citation
 PubChem, PC Dose Response with BCECF Assay for V-ATPase inhibitors that increase vacuolar pH, Powder Set 1 PubChem Bioassay (2012)[AID] 
Target
Name:
V-type proton ATPase subunit c'
Synonyms:
CLS9 | TFP3 | VATL2_YEAST | VMA11 | Vma11p
Type:
Enzyme Catalytic Domain
Mol. Mass.:
17039.28
Organism:
Saccharomyces cerevisiae S288c
Description:
gi_6325022
Residue:
164
Sequence:
MSTQLASNIYAPLYAPFFGFAGCAAAMVLSCLGAAIGTAKSGIGIAGIGTFKPELIMKSLIPVVMSGILAIYGLVVAVLIAGNLSPTEDYTLFNGFMHLSCGLCVGFACLSSGYAIGMVGDVGVRKYMHQPRLFVGIVLILIFSEVLGLYGMIVALILNTRGSE
  
Inhibitor
Name:
BDBM3738
Synonyms:
cid_32250470
Type:
n/a
Emp. Form.:
C15H13F3N4O4
Mol. Mass.:
370.2833
SMILES:
[O-][N+](=O)c1ccc(o1)C(=O)N1CCN(CC1)c1ccc(cn1)C(F)(F)F
Structure:
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