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Target
Mitochondrial peptide methionine sulfoxide reductase
Ligand
BDBM91499
Substrate
n/a
Meas. Tech.
Absorbance-based biochemical high throughput dose response assay for activators of Methionine sulfoxide reductase A (MsrA)
EC50
>103851±n/a nM
Citation
 PubChem, PC Absorbance-based biochemical high throughput dose response assay for activators of Methionine sulfoxide reductase A (MsrA) PubChem Bioassay (2012)[AID] 
Target
Name:
Mitochondrial peptide methionine sulfoxide reductase
Synonyms:
MSRA | MSRA protein | MSRA_BOVIN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
25822.90
Organism:
Bos taurus
Description:
gi_73586699
Residue:
233
Sequence:
MLSATRRALQLFHSLFPIPRMGDSAAKIVSPQEALPGRKEPLVVAAKHHVNGNRTVEPFPEGTQMAVFGMGCFWGAERKFWTLKGVYSTQVGFAGGYTPNPTYKEVCSGKTGHAEVVRVVFQPEHISFEELLKVFWENHDPTQGMRQGNDHGSQYRSAIYPTSAEHVGAALKSKEDYQKVLSEHGFGLITTDIREGQTFYYAEDYHQQYLSKDPDGYCGLGGTGVSCPLGIKK
  
Inhibitor
Name:
BDBM91499
Synonyms:
(3-amino-5,8-dimethyl-2-thieno[2,3-b]quinolinyl)-(4-morpholinyl)methanone | (3-amino-5,8-dimethyl-thieno[2,3-b]quinolin-2-yl)-morpholino-methanone | (3-amino-5,8-dimethylthieno[2,3-b]quinolin-2-yl)-morpholin-4-ylmethanone | (3-azanyl-5,8-dimethyl-thieno[2,3-b]quinolin-2-yl)-morpholin-4-yl-methanone | MLS000692916 | SMR000285651 | cid_865023
Type:
Small organic molecule
Emp. Form.:
C18H19N3O2S
Mol. Mass.:
341.427
SMILES:
Cc1ccc(C)c2nc3sc(C(=O)N4CCOCC4)c(N)c3cc12
Structure:
Search PDB for entries with ligand similarity: