Reaction Details Report a problem with these data
Target
Heat shock protein hsp-16.2
Ligand
BDBM93917
Substrate
n/a
IC50
>64000±n/a nM
Citation
 PubChem, PC Dose Response Confirmation of SKN-1 Inhibitor hits via a heat-shock counterscreen assay PubChem Bioassay (2012)[AID] 
Target
Name:
Heat shock protein hsp-16.2
Synonyms:
HSP12_CAEEL | Protein HSP-16.2 | hsp-16 | hsp-16.2 | hsp16-2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
16239.18
Organism:
Caenorhabditis elegans
Description:
gi_373219859
Residue:
145
Sequence:
MSLYHYFRPAQRSVFGDLMRDMALMERQFAPVCRISPSESSEIVNNDQKFAINLNVSQFKPEDLKINLDGRTLSIQGEQELKTDHGYSKKSFSRVILLPEDVDVGAVASNLSEDGKLSIEAPKKEAVQGRSIPIQQAIVEEKSAE
  
Inhibitor
Name:
BDBM93917
Synonyms:
5-(4-morpholinyl)-1,5-diphenyl-1-penten-3-one | 5-morpholin-4-yl-1,5-diphenyl-pent-1-en-3-one | 5-morpholin-4-yl-1,5-diphenylpent-1-en-3-one | 5-morpholino-1,5-diphenyl-pent-1-en-3-one | MLS002639478 | SMR001548922 | cid_234165
Type:
Small organic molecule
Emp. Form.:
C21H23NO2
Mol. Mass.:
321.4128
SMILES:
O=C(CC(N1CCOCC1)c1ccccc1)C=Cc1ccccc1 |w:16.17|
Structure:
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