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Targetperilipin-5
LigandBDBM70875
Substrate/Competitorn/a
IC50 1705±n/a nM
Citation PubChem, PC Luminescence-based biochemical high throughput dose response assay for inhibitors of the interaction of the lipase co-activator protein, abhydrolase domain containing 5 (ABHD5) with perilipin-5 (MLDP; PLIN5) produced in HEK293T cells PubChem Bioassay(2012)[AID]
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perilipin-5
Name:perilipin-5
Synonyms:n/a
Type:Enzyme Catalytic Domain
Mol. Mass.:50774.20
Organism:Homo sapiens (Human)
Description:gi_116292172
Residue:463
Sequence:
MSEEEAAQIPRSSVWEQDQQNVVQRVVALPLVRATCTAVCDVYSAAKDRHPLLGSACRLA
ENCVCGLTTRALDHAQPLLEHLQPQLATMNSLACRGLDKLEEKLPFLQQPSETVVTSAKD
VVASSVTGVVDLARRGRRWSVELKRSVSHAVDVVLEKSEELVDHFLPMTEEELAALAAEA
EGPEVGSVEDQRRQQGYFVRLGSLSARIRHLAYEHSVGKLRQSKHRAQDTLAQLQETLEL
IDHMQCGVTPTAPACPGKVHELWGEWGQRPPESRRRSQAELETLVLSRSLTQELQGTVEA
LESSVRGLPAGAQEKVAEVRRSVDALQTAFADARCFRDVPAAALAEGRGRVAHAHACVDE
LLELVVQAVPLPWLVGPFAPILVERPEPLPDLADLVDEVIGGPDPRWAHLDWPAQQRAWE
AEHRDGSGNGDGDRMGVAGDICEQEPETPSCPVKHTLMPELDF
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  Blast E-value cutoff:
BDBM70875
NameBDBM70875
Synonyms:(Z)-2-(1,3-benzothiazol-2-yl)-N-(4-chlorophenyl)-3-(3-hydroxyphenyl)-2-propenamide | (Z)-2-(1,3-benzothiazol-2-yl)-N-(4-chlorophenyl)-3-(3-hydroxyphenyl)acrylamide | (Z)-2-(1,3-benzothiazol-2-yl)-N-(4-chlorophenyl)-3-(3-hydroxyphenyl)prop-2-enamide | MLS000392964 | SMR000248103 | cid_8259799
TypeSmall organic molecule
Emp. Form.C22H15ClN2O2S
Mol. Mass.406.885
SMILESOc1cccc(\C=C(\C(=O)Nc2ccc(Cl)cc2)c2nc3ccccc3s2)c1
Structure
n/a