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Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM96748
Substrate
n/a
EC50
>29887±n/a nM
Citation
 PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 agonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | guanine nucleotide-binding protein subunit alpha-15
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Homo sapiens (Human)
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRAYYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM96748
Synonyms:
(4-aminoquinazolin-2-yl)-(3,4-dimethylphenyl)amine;hydrochloride | 2-N-(3,4-dimethylphenyl)quinazoline-2,4-diamine;hydrochloride | MLS001001860 | N2-(3,4-dimethylphenyl)quinazoline-2,4-diamine;hydrochloride | N~2~-(3,4-dimethylphenyl)-2,4-quinazolinediamine hydrochloride | SMR000498358 | cid_2975866
Type:
Small organic molecule
Emp. Form.:
C16H16N4
Mol. Mass.:
264.325
SMILES:
Cc1ccc(Nc2nc(N)c3ccccc3n2)cc1C
Structure:
Search PDB for entries with ligand similarity: