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Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM96606
Substrate
n/a
IC50
29775±n/a nM
Citation
 PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 antagonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | guanine nucleotide-binding protein subunit alpha-15
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Homo sapiens (Human)
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRAYYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM96606
Synonyms:
1-(4-acetylphenyl)-3-phenyl-urea | 1-(4-acetylphenyl)-3-phenylurea | 1-(4-ethanoylphenyl)-3-phenyl-urea | MLS000532118 | N-(4-acetylphenyl)-N'-phenylurea | SMR000137059 | cid_682184
Type:
Small organic molecule
Emp. Form.:
C15H14N2O2
Mol. Mass.:
254.2839
SMILES:
CC(=O)c1ccc(NC(=O)Nc2ccccc2)cc1
Structure:
Search PDB for entries with ligand similarity: