Reaction Details Report a problem with these data
Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM96911
Substrate
n/a
EC50
>29910±n/a nM
Citation
 PubChem, PC Counterscreen for antagonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose reponse assay to identify nonselective Ga16 agonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | guanine nucleotide-binding protein subunit alpha-15
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Homo sapiens (Human)
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRAYYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM96911
Synonyms:
2-(3-bromobenzyl)oxy-N-[(E)-(5-methyl-2-furyl)methyleneamino]benzamide | 2-[(3-bromobenzyl)oxy]-N'-[(1E)-(5-methyl-2-furyl)methylene]benzohydrazide | 2-[(3-bromophenyl)methoxy]-N-[(E)-(5-methyl-2-furanyl)methylideneamino]benzamide | 2-[(3-bromophenyl)methoxy]-N-[(E)-(5-methylfuran-2-yl)methylideneamino]benzamide | MLS000723745 | SMR000305340 | cid_46497982
Type:
Small organic molecule
Emp. Form.:
C20H17BrN2O3
Mol. Mass.:
413.265
SMILES:
Cc1ccc(\C=N\NC(=O)c2ccccc2OCc2cccc(Br)c2)o1
Structure:
Search PDB for entries with ligand similarity: