Reaction Details Report a problem with these data
Target
Galanin receptor type 3
Ligand
BDBM89372
Substrate
n/a
IC50
140.16±n/a nM
Citation
 PubChem, PC Fluorescence-based cell-based primary high throughput dose response assay to identify antagonists of the Galanin Receptor 3 (GalR3). PubChem Bioassay (2013)[AID] 
Target
Name:
Galanin receptor type 3
Synonyms:
GALNR3 | GALR3 | GALR3_HUMAN | Galanin R3 | Galanin receptor 3 | Galanin receptor type 3
Type:
Enzyme Catalytic Domain
Mol. Mass.:
39599.97
Organism:
Homo sapiens (Human)
Description:
Galanin R3 GALR3 HUMAN::O60755
Residue:
368
Sequence:
MADAQNISLDSPGSVGAVAVPVVFALIFLLGTVGNGLVLAVLLQPGPSAWQEPGSTTDLFILNLAVADLCFILCCVPFQATIYTLDAWLFGALVCKAVHLLIYLTMYASSFTLAAVSVDRYLAVRHPLRSRALRTPRNARAAVGLVWLLAALFSAPYLSYYGTVRYGALELCVPAWEDARRRALDVATFAAGYLLPVAVVSLAYGRTLRFLWAAVGPAGAAAAEARRRATGRAGRAMLAVAALYALCWGPHHALILCFWYGRFAFSPATYACRLASHCLAYANSCLNPLVYALASRHFRARFRRLWPCGRRRRHRARRALRRVRPASSGPPGCPGDARPSGRLLAGGGQGPEPREGPVHGGEAARGPE
  
Inhibitor
Name:
BDBM89372
Synonyms:
1-(4-bromobenzyl)-2-methyl-1H-benzimidazole | 1-(4-bromobenzyl)-2-methyl-benzimidazole | 1-[(4-bromophenyl)methyl]-2-methyl-benzimidazole | 1-[(4-bromophenyl)methyl]-2-methylbenzimidazole | MLS001077238 | SMR000473021 | cid_743662
Type:
Small organic molecule
Emp. Form.:
C15H13BrN2
Mol. Mass.:
301.181
SMILES:
Cc1nc2ccccc2n1Cc1ccc(Br)cc1
Structure:
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