Target
5-hydroxytryptamine 1D receptor
Ligand
BDBM106703
Substrate
n/a
Meas. Tech.
Binding Assay
IC50
8.7e+2±n/a nM
Citation
 Maddaford, SRamnauth, JRakhit, SPatman, JRenton, PAnnedi, SC Substituted indole compounds having NOS inhibitory activity US Patent  US8586620 Publication Date 11/19/2013 
Target
Name:
5-hydroxytryptamine 1D receptor
Synonyms:
5-hydroxytryptamine 1D receptor (5HT1D) | HTR1D
Type:
Protein
Mol. Mass.:
12731.52
Organism:
Bos taurus (Bovine)
Description:
Q8MI13
Residue:
119
Sequence:
SNRSLNATATQGAWDPGTLQALKIALVVLLSIITLATVLSNAFVLTTIFLTRKLHTPANCLIGSLAMTDLLVSILVMPISIAYTTTHTWSFGQLLCDIWLSSDITCCTASILHLCVIAL
  
Inhibitor
Name:
BDBM106703
Synonyms:
US8586620, 15
Type:
Small organic molecule
Emp. Form.:
C18H22N4S
Mol. Mass.:
326.459
SMILES:
CN(C)CCCc1c[nH]c2ccc(cc12)N=C(N)c1cccs1 |w:15.16|
Structure:
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