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Target
ELAV-like protein 1 [I180A]
Ligand
BDBM128146
Substrate
n/a
IC50
26900±n/a nM
Citation
 PubChem, PC Identify HuR specific inhibitors PubChem Bioassay (2015)[AID] 
Target
Name:
ELAV-like protein 1 [I180A]
Synonyms:
ELAV1_HUMAN | ELAVL1 | HUR | HuR RNA binding protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
36072.53
Organism:
Homo sapiens (Human)
Description:
gi_1022961
Residue:
326
Sequence:
MSNGYEDHMAEDCRGDIGRTNLIVNYLPQNMTQDELRSLFSSIGEVESAKLIRDKVAGHSLGYGFVNYVTAKDAERAINTLNGLRLQSKTIKVSYARPSSEVIKDANLYISGLPRTMTQKDVEDMFSRFGRIINSRVLVDQTTGLSRGVAFIRFDKRSEAEEAITSFNGHKPPGSSEPIAVKFAANPNQNKNVALLSQLYHSPARRFGGPVHHQAQRFRFSPMGVDHMSGLSGVNVPGNASSGWCIFIYNLGQDADEGILWQMFGPFGAVTNVKVIRDFNTNKCKGFGFVTMTNYEEAAMAIASLNGYRLGDKILQVSFKTNKSHK
  
Inhibitor
Name:
BDBM128146
Synonyms:
3,5-bis(2,5-dioxo-1-pyrrolyl)benzoic acid | 3,5-bis(2,5-dioxopyrrol-1-yl)benzoic acid | 3,5-bis[2,5-bis(oxidanylidene)pyrrol-1-yl]benzoic acid | 3,5-dimaleimidobenzoic acid | MLS002608658 | SMR001527404 | cid_239577
Type:
Small organic molecule
Emp. Form.:
C15H8N2O6
Mol. Mass.:
312.2338
SMILES:
OC(=O)c1cc(cc(c1)N1C(=O)C=CC1=O)N1C(=O)C=CC1=O |c:13,21|
Structure:
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