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Target
ELAV-like protein 1 [I180A]
Ligand
BDBM200226
Substrate
n/a
IC50
21700±n/a nM
Citation
 PubChem, PC Identify HuR specific inhibitors PubChem Bioassay (2015)[AID] 
Target
Name:
ELAV-like protein 1 [I180A]
Synonyms:
ELAV1_HUMAN | ELAVL1 | HUR | HuR RNA binding protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
36072.53
Organism:
Homo sapiens (Human)
Description:
gi_1022961
Residue:
326
Sequence:
MSNGYEDHMAEDCRGDIGRTNLIVNYLPQNMTQDELRSLFSSIGEVESAKLIRDKVAGHSLGYGFVNYVTAKDAERAINTLNGLRLQSKTIKVSYARPSSEVIKDANLYISGLPRTMTQKDVEDMFSRFGRIINSRVLVDQTTGLSRGVAFIRFDKRSEAEEAITSFNGHKPPGSSEPIAVKFAANPNQNKNVALLSQLYHSPARRFGGPVHHQAQRFRFSPMGVDHMSGLSGVNVPGNASSGWCIFIYNLGQDADEGILWQMFGPFGAVTNVKVIRDFNTNKCKGFGFVTMTNYEEAAMAIASLNGYRLGDKILQVSFKTNKSHK
  
Inhibitor
Name:
BDBM200226
Synonyms:
cid_83851
Type:
Small organic molecule
Emp. Form.:
C27H30N2O10
Mol. Mass.:
542.5345
SMILES:
COc1cccc2C(=O)c3c(O)c4CC(O)(CC(OC5CC(N)C(O)C(C)O5)c4c(O)c3C(=O)c12)C(C)=NO
Structure:
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