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Target
ELAV-like protein 1 [I180A]
Ligand
BDBM200227
Substrate
n/a
IC50
17400±n/a nM
Citation
 PubChem, PC Identify HuR specific inhibitors PubChem Bioassay (2015)[AID] 
Target
Name:
ELAV-like protein 1 [I180A]
Synonyms:
ELAV1_HUMAN | ELAVL1 | HUR | HuR RNA binding protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
36072.53
Organism:
Homo sapiens (Human)
Description:
gi_1022961
Residue:
326
Sequence:
MSNGYEDHMAEDCRGDIGRTNLIVNYLPQNMTQDELRSLFSSIGEVESAKLIRDKVAGHSLGYGFVNYVTAKDAERAINTLNGLRLQSKTIKVSYARPSSEVIKDANLYISGLPRTMTQKDVEDMFSRFGRIINSRVLVDQTTGLSRGVAFIRFDKRSEAEEAITSFNGHKPPGSSEPIAVKFAANPNQNKNVALLSQLYHSPARRFGGPVHHQAQRFRFSPMGVDHMSGLSGVNVPGNASSGWCIFIYNLGQDADEGILWQMFGPFGAVTNVKVIRDFNTNKCKGFGFVTMTNYEEAAMAIASLNGYRLGDKILQVSFKTNKSHK
  
Inhibitor
Name:
BDBM200227
Synonyms:
cid_374010
Type:
Small organic molecule
Emp. Form.:
C16H17N3O6
Mol. Mass.:
347.3227
SMILES:
COCC(=O)OC1CCn2c1nc1c2C(=O)C(C)=C(NC(C)=O)C1=O |t:19|
Structure:
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