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Target
DNA-directed RNA polymerase subunit alpha
Ligand
BDBM466508
Substrate
n/a
Meas. Tech.
Assay of Inhibition of Staphylococcus Aureus RNA Polymerase
IC50
>400000±n/a nM
Citation
Ebright, RH; Shen, J Arylpropionyl-triketone antibacterial agents US Patent US10800725 Publication Date 10/13/2020
More Info.:
Target
Name:
DNA-directed RNA polymerase subunit alpha
Synonyms:
RNA polymerase subunit alpha | RNAP subunit alpha | RPOA_STAAN | Transcriptase subunit alpha | rpoA
Type:
Protein
Mol. Mass.:
34991.14
Organism:
n/a
Description:
P66706
Residue:
314
Sequence:
MIEIEKPRIETIEISEDAKFGKFVVEPLERGYGTTLGNSLRRILLSSLPGAAVKYIEIEGVLHEFSAVDNVVEDVSTIIMNIKQLALKIYSEEDKTLEIDVRDEGEVTASDITHDSDVEILNPELKIATVSKGGHLKIRLVANKGRGYALAEQNNTSDLPIGVIPVDSLYSPVERVNYTVENTRVGQSSDFDKLTLDVWTNGSITPQESVSLAAKIMTEHLNIFVGLTDEAQNAEIMIEKEEDQKEKVLEMSIEELDLSVRSYNCLKRAGINSVQELADKSEADMMKVRNLGRKSLEEVKYKLEDLGLGLRKED