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Target
Resistin
Ligand
BDBM486500
Substrate
n/a
Meas. Tech.
Evaluation of the Ability to Inhibit TNF-α Secretion by human Resistin
IC50
7900±n/a nM
Citation
 Yoo, JK; Lee, N; Lee, CH; Jung, M; Kim, H Phenyl phthalazine derivative, method for the preparation thereof, and pharmaceutical composition comprising the same US Patent  US10947241 Publication Date 3/16/2021 
Target
Name:
Resistin
Synonyms:
ADSF | Adipose tissue-specific secretory factor | C/EBP-epsilon-regulated myeloid-specific secreted cysteine-rich protein | Cysteine-rich secreted protein A12-alpha-like 2 | Cysteine-rich secreted protein FIZZ3 | FIZZ3 | HXCP1 | RETN | RETN_HUMAN | RSTN
Type:
Protein
Mol. Mass.:
11419.78
Organism:
Human
Description:
Q9HD89
Residue:
108
Sequence:
MKALCLLLLPVLGLLVSSKTLCSMEEAINERIQEVAGSLIFRAISSIGLECQSVTSRGDLATCPRGFAVTGCTCGSACGSWDVRAETTCHCQCAGMDWTGARCCRVQP
  
Inhibitor
Name:
BDBM486500
Synonyms:
US10947241, Example 38
Type:
Small organic molecule
Emp. Form.:
C20H22ClN5
Mol. Mass.:
367.875
SMILES:
NCCN1CCN(CC1)c1nnc(-c2ccc(Cl)cc2)c2ccccc12
Structure:
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