Assay Method Information

Assay Name:  ChEMBL_1654441 (CHEMBL4003807)
Description:  Antagonist activity at human adenosine A2A receptor expressed in HEK293 cell membranes assessed as decrease in CGS-21680/forskolin-induced cAMP level pretreated for 15 mins followed by agonist addition for 30 mins and subsequent forskolin stimulation measured after 30 mins
Affinity data for this assay
 

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