Assay Method Information | |
| ChEMBL_2059672 (CHEMBL4714673) |
Description: | Orthosteric agonist activity at recombinant human N-terminal His6-tagged RORgammat ligand binding domain (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as increase in coactivator, N-terminal biotinylated SRC-1 box2 peptide recruitment incubated for 60 mins by TR-FRET assay |
Affinity data for this assay | |
---|---|
If you find an error in this entry please send us an E-mail |