Assay Method Information

Assay Name:  ChEMBL_2059672 (CHEMBL4714673)
Description:  Orthosteric agonist activity at recombinant human N-terminal His6-tagged RORgammat ligand binding domain (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as increase in coactivator, N-terminal biotinylated SRC-1 box2 peptide recruitment incubated for 60 mins by TR-FRET assay
Affinity data for this assay
 

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