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26 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Systemic optimization and structural evaluation of quinoline derivatives as transthyretin amyloidogenesis inhibitors.EBI
Chungnam National University
A novel bis-furan scaffold for transthyretin stabilization and amyloid inhibition.EBI
Universidade De Coimbra
Enthalpic Forces Correlate with the Selectivity of Transthyretin-Stabilizing Ligands in Human Plasma.EBI
Ume£
Inhibitory activities of propolis and its promising component, caffeic acid phenethyl ester, against amyloidogenesis of human transthyretin.EBI
University Of Toyama
Synthesis and evaluation of transthyretin amyloidosis inhibitors containing carborane pharmacophores.EBI
University Of California
Chemoselective small molecules that covalently modify one lysine in a non-enzyme protein in plasma.EBI
The Scripps Research Institute
Identification of a novel ligand binding motif in the transthyretin channel.EBI
Universidade Federal Do Rio De Janeiro
Isatin derivatives, a novel class of transthyretin fibrillogenesis inhibitors.EBI
Universitat De Barcelona
Design of mechanism-based inhibitors of transthyretin amyloidosis: studies with biphenyl ethers and new structural templates.EBI
Institute Of Sciences
Repositioning of the Anthelmintic Drugs Bithionol and Triclabendazole as Transthyretin Amyloidogenesis Inhibitors.EBI
University Of Toyama
Inhibitory activities of anthraquinone and xanthone derivatives against transthyretin amyloidogenesis.EBI
University Of Toyama
Transthyretin Amyloidogenesis Inhibitors: From Discovery to Current Developments.EBI
University Of Toyama
Discovery of Bispecific Antagonists of Retinol Binding Protein 4 That Stabilize Transthyretin Tetramers: Scaffolding Hopping, Optimization, and Preclinical Pharmacological Evaluation as a Potential Therapy for Two Common Age-Related Comorbidities.EBI
Albany College Of Pharmacy And Health Sciences
Crown Ethers as Transthyretin Amyloidogenesis Inhibitors.EBI
University Of Toyama
Calorimetric Studies of Binary and Ternary Molecular Interactions between Transthyretin, A? Peptides, and Small-Molecule Chaperones toward an Alternative Strategy for Alzheimer's Disease Drug Discovery.EBI
Institut De Qu??Mica Avan£Ada De Catalunya (I.Q.A.C.-C.S.I.C.)
Enthalpy-Driven Stabilization of Transthyretin by AG10 Mimics a Naturally Occurring Genetic Variant That Protects from Transthyretin Amyloidosis.EBI
University Of The Pacific
Insights on the Interaction between Transthyretin and A? in Solution. A Saturation Transfer Difference (STD) NMR Analysis of the Role of Iododiflunisal.EBI
Cic Biogune
Stilbene Boronic Acids Form a Covalent Bond with Human Transthyretin and Inhibit Its Aggregation.EBI
University Of Wisconsin-Madison
Carbonic anhydrase inhibitory properties of novel sulfonamide derivatives of aminoindanes and aminotetralins.BDB
Atatürk University
Peripheral-type benzodiazepine receptors in human cerebral cortex, kidney, and colon.BDB
Technion-Israel Institute Of Technology
Carbonic anhydrase inhibitors: stacking with Phe131 determines active site binding region of inhibitors as exemplified by the X-ray crystal structure of a membrane-impermeant antitumor sulfonamide complexed with isozyme II.BDB
Istituto Di Biostrutture E Bioimmagini-Cnr